Pharmacological and molecular studies on the interaction of varenicline with different nicotinic acetylcholine receptor subtypes. Potential mechanism underlying partial agonism at human α4β2 and α3β4 subtypes
Keywords: nAChR; nicotinic acetylcholine receptor; [3H]MLA; [3H]methyllycaconitine; [3H]TCP; piperidyl-3, 4-3H(N)]-(N-(1-(2 thienyl)cyclohexyl)-3, 4-piperidine; α-BTx; α-bungarotoxin; Varenicline; 7,8,9,10-tetrahydro-6,10-methano-6H-azepino[4,5-g]quinoxaline; RT;